找到约 38 条 “Compound E” 相关结果 (用时 0.178 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M2238 | Dorsomorphin (Compound C) dihydrochloride | Dorsomorphin (Compound C) dihydrochloride | AMPK |
BML-275 2HCl; Compound C 2HCl | |||
Dorsomorphin (BML-275)二盐酸盐是一种有效的,可逆的AMPK选择性抑制剂,Ki为109 nM,Dorsomorphin还对BMP有抑制作用。 | |||
M5534 | Cortisone | 可的松 | GCR |
17-Hydroxy-11-dehydrocorticosterone; Kendall's compound E | |||
Cortisone是一种用于治疗感染或过敏的激素药物 | |||
M7043 | NPS ALX Compound 4a dihydrochloride | NPS ALX Compound 4a dihydrochloride | Others |
NPS ALX Compound 4a dihydrochloride is a potent and selective 5-HT 6 antagonist. | |||
M9505 | Compound E | Compound E | Gamma-secretase/Beta-secretase |
GSI-XXI; γ-secretase inhibitor XXI; γ-Secretase-IN-1 | |||
Compound E 是一种可透过细胞的强效选择性γ-分泌酶(γ-secretase)和Notch抑制剂。 | |||
M11655 | ChemBridge-5126190 | ChemBridge化合物-5126190 | Screening Compounds and Building Blocks |
3,7-dihydro-1H-purine-2,6-dione (5126190) | |||
ChemBridge特有类药化合物/先导化合物-5126190,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12301 | ChemBridge-5713492 | ChemBridge化合物-5713492 | Screening Compounds and Building Blocks |
1-(2-chloro-4-nitrophenyl)-4-[(5-methyl-3-phenyl-4-isoxazolyl)carbonyl]piperazine (5713492) | |||
ChemBridge特有类药化合物/先导化合物-5713492,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12806 | ChemBridge-6881166 | ChemBridge化合物-6881166 | Screening Compounds and Building Blocks |
4-[(2-{[1-(4-ethylphenyl)-2,4,6-trioxotetrahydro-5(2H)-pyrimidinylidene]methyl}phenoxy)methyl]benzoic acid (6881166) | |||
ChemBridge特有类药化合物/先导化合物-6881166,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M20547 | Rabeprazole Related Compound E | Rabeprazole Related Compound E | Proton Pump |
Rabeprazole thioether; Rabeprazole Sulfide | |||
Rabeprazole Related Compound E是 Rabeprazole 的活性代谢产物,同时也是一种具有口服活性的质子泵抑制剂,能通过与胃壁细胞中的 (H+/K+)-ATPase 相互作用来抑制胃酸分泌。此外,Rabeprazole Related Compound E 还能显著抑制幽门螺旋杆菌的活性,可用于各种消化系统疾病的相关研究。 | |||
M20688 | B-Raf inhibitor 1 (Compound 13) dihydrochloride | B-Raf inhibitor 1 (Compound 13) dihydrochloride | Raf |
B-Raf inhibitor 1 (Compound 13) is a type IIA Raf inhibitor which bind to the DFG-out conformation with ki of 1 nM,1 nM,and 0.3 nM for B-Raf(WT), B-Raf(V600E) and C-Raf, respectively. | |||
M21681 | Compound 48/80 trihydrochloride | Compound 48/80 trihydrochloride | Phospholipase |
C48/80 trihydrochloride | |||
Compound 48/80 trihydrochloride 作为选择性肥大细胞激活剂广泛用于动物和组织模型。Compound 48/80 作用于肥大细胞膜,刺激三聚体 G 蛋白,并通过磷脂酶 C 和 D 途径诱导脱颗粒。 | |||
M2608 | Kobe0065 | Kobe0065 | Ras |
Kobe0065 is a novel and effective small-molecule compound inhibiting Ras–Raf interaction by SBDD, exhibits potent activity to competitively inhibit the binding of H-Ras·GTP to c-Raf-1 RBD with a Ki value of 46 ± 13 μM. | |||
M2896 | OAC1 | OAC1 | Others |
OAC1 (Oct4-activating compound 1)是一种有效的 Oct4 激活剂,能激活 Oct4 和 Nanog 启动子,促进诱导多功能干细胞 (iPSC) 的形成,以及通过上调 HOXB4 表达激活 OCT4。此外,OAC1 还能增加Oct4-Nanog-Sox2 三联体和 TET1 的转录,并可通过提高效率和缩短重编程时间,促进细胞的重编程。 | |||
M4088 | Ginsenoside Compound-K | 人参皂苷CK | COX |
Ginsenoside K; Ginsenoside C-K | |||
Ginsenoside Compound-K(人参皂苷CK)是一种 Ginsenoside Rb1 细菌代谢物,通过抑制诱生型一氧化氮合酶 (iNOS) 和 COX-2,从而发挥抗炎作用。 | |||
M4902 | Chloroxine | 克氯辛;氯喔星 | Antibiotic |
Chloroxine is a synthetic antibacterial compound that is effective in the treatment of dandruff and seborrheic dermatitis when incorporated in a shampoo. | |||
M4924 | Dehydroacetic acid | 脱氢乙酸 | Antibiotic |
Biocide 470F | |||
Dehydroacetic acid is an organic compound, classified as a pyrone derivative and is used mostly as a fungicide and bactericide. | |||
M4961 | CB72666407 | CB72666407 | mTOR |
Pyrimidine substituted purine compounds as kinase (S) inhibitors. | |||
M4987 | Procyanidin B4 | Procyanidin B4 | Others |
A series of dimeric procyanidins (1-9) and some related polyphenols (10-15) were chosen as model compounds in a comparative investigation for various biological activities in order to obtain structure-activity relationships. | |||
M5007 | Hexyl Chloroformate | 己基甲酸氯 | Others |
The Carbonochloridic acid,hexyl ester, belongs to the following product categories: (1)Acid Halides; (2)Carbonyl Compounds; (3)Organic Building Blocks. It has the systematic name of hexyl carbonochloridate. | |||
M6285 | Glutaminase C-IN-1 | Glutaminase C-IN-1 | Glutaminase |
Compound 968 | |||
Glutaminase C-IN-1 (Compound 968) 是一种Glutaminase C变构抑制剂。 | |||
M7400 | Teijin compound 1 | Teijin compound 1 | Others |
Teijin compound 1 is a potent CCR2b antagonist. | |||
M7838 | 8-Hydroxy-2′-deoxyguanosine | 8-Hydroxy-2′-deoxyguanosine | Metabolite/Endogenous Metabolite |
A marker compound typically indicative of DNA damage associated with mutagenesis and carcinogenesis. | |||
M7946 | Naloxone methiodide | Naloxone methiodide | Others |
Quaternary salt of naloxone that, like the parent compound, is a nonselective antagonist at opioid receptors. | |||
M8161 | SE 175 | SE 175 | Others |
An organic nitrate compound that acts as an NO donor in vivo following reductive transformation of the nitrate group to nitric oxide. | |||
M8166 | Sulindac sulfide | 硫化舒林酸 | Others |
Sulindac sulfide is a non-steroidal anti-inflammatory compound with a preference for COX-1; it is an inhibitor of Ras activation of Raf-1. | |||
M8211 | Triacetyl resveratrol | 乙酰化白藜芦醇 | STAT |
Triacetyl resveratrol displays superior bioavailability to the parent compound, resveratrol. | |||
M8246 | GPR35 Agonist, Compound 10 | GPR35 Agonist, Compound 10 | Others |
GPR35 agonist Compound 10 is a GPR35 agonist the binds with higher affinity than other known agonists, such as kynurenic acid and zaprinast. | |||
M8609 | MM-206 | MM-206 | Others |
MM-206 is a cell-permeable, non-cytotoxic naphthalene sulfonamide compound effectively inhibits STAT3 DNA-binding activity (IC50 = 2. | |||
M8635 | Displurigen | Displurigen | Others |
Displurigen is a cell-permeable, phenylthiochromen-4-one derived compound that disrupts the pluripotency of human embryonic stem cells by targeting HSPA8/HSC70 and affects its binding to Oct4. | |||
M8639 | STK16-IN-1 | STK16-IN-1 | Others |
STK16-IN-1 is a cell-permeable pyrrolonaphthyridinone compound that acts as an ATP-competitive inhibitor against NAK (Numb Associated Kinase) family serine/threonine kinase STK16 (IC50/substrate = 0. | |||
M8640 | SW044248 | SW044248 | Topoisomerase |
SW044248 is a cell permeable, indolotriazine-based compound that selectively inhibits topoisomerase 1 (Top 1), but not Top 2, catalyzed DNA decatenation in a manner distinct from that of camptothecin (Cat. | |||
M8647 | Raptinal | Raptinal | Caspase |
Raptinal is a cell-permeable bifluorene-dicarbaldehyde compound that acts as a rapid activator of mitochondrial pathway-mediated intrinsic apoptosis. | |||
M8668 | MI-4F | MI-4F | Others |
MI-4F is mesoionic compound that exhibits potent anticancer activity against multiple cancer cell lines and in vivo. | |||
M8706 | NSC57969 | NSC57969 | Others |
NSC57969 is a MDR-selective compound that exhibits a robust Pgp-dependent toxic activity across diverse cancer cell lines. | |||
M8717 | PBOX-6 | PBOX-6 | Others |
PBOX-6 belongs to a group of tubulin-targeting pyrrolo-1,5-benzoxazepine (PBOX) compounds that potently induce apoptosis in a wide spectrum of cancer cells, including those originating from the four main types of leukemia. | |||
M8723 | PBOX-15 | PBOX-15 | Others |
PBOX-15 belongs to a group of tubulin-targeting pyrrolo-1,5-benzoxazepine (PBOX) compounds that potently induce apoptosis in a wide spectrum of cancer cells, including those originating from the four main types of leukemia. | |||
M8884 | Febantel | 非班太尔 | Parasite |
Rintal, Combotel | |||
Febantel is a veteran anthelmintic (wormer) compound belonging to the chemical class of the benzimidazoles. | |||
M9031 | 6-Methylcoumarin | 6-Methylcoumarin | Others |
Toncarine | |||
6-Methylcoumarin belongs to the class of organic compounds known as coumarins and derivatives. | |||
M9461 | Oxyclozanide | 氯羟柳胺;五氯柳胺;羟氯柳苯胺 | Anti-infection |
五氯柳胺Oxyclozanide is a salicylanilide anthelmintic compound, which acts by uncoupling oxidative phosphorylation in flukes. |
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